DRUGS sens assoc res assoc tot 1378 - Bleomycin (50 uM) [DNA damage] 1 17 18 1047 - Nutlin-3a [MDM2] 1 14 15 208 - SB-715992 [KIF11] 1 10 11 1175 - AG-014699 [PARP1, PARP2] 1 8 9 179 - 5-Fluorouracil [DNA antimetabolite] 0 9 9 300 - CX-5461 [RNA Pol I] 3 6 9 1003 - Camptothecin [TOP1] 1 6 7 1054 - PD-0332991 [CDK4, CDK6] 1 6 7 1012 - Vorinostat [HDAC inhibitor Class I, IIa, IIb, IV] 0 6 6 1239 - YK 4-279 [RNA helicase A] 0 6 6 257 - NPK76-II-72-1 [PLK3] 2 4 6 1009 - ATRA [Retinoic acid and retinoid X receptor agonist] 2 3 5 1014 - RDEA119 [MAP2K1 (MEK1), MAP2K2 (MEK2)] 4 1 5 1015 - CI-1040 [MAP2K1 (MEK1), MAP2K2 (MEK2)] 3 2 5 1050 - ZM-447439 [AURKB] 1 4 5 1057 - NVP-BEZ235 [PI3K (Class 1) and MTORC1/2] 0 5 5 110 - Roscovitine [CDKs] 0 5 5 1129 - PF-4708671 [RPS6KB1 (p70S6KA)] 0 5 5 1242 - (5Z)-7-Oxozeaenol [MAP3K7 (TAK1)] 1 4 5 1498 - AZD6244 [MAP2K1 (MEK1), MAP2K2 (MEK2)] 4 1 5 1526 - RDEA119 (rescreen) [MAP2K1 (MEK1), MAP2K2 (MEK2)] 3 2 5 230 - GSK429286A [ROCK2] 5 0 5 272 - AR-42 [HDAC] 1 4 5 290 - KIN001-260 [IKK] 3 2 5 326 - GSK690693 [AKT] 5 0 5 330 - XMD13-2 [RIPK] 2 3 5 1013 - Nilotinib [ABL] 4 0 4 1021 - Axitinib [PDGFR, KIT, VEGFR] 3 1 4 1024 - CEP-701 [FLT3, JAK2, NTRK1, RET] 0 4 4 1049 - PD-173074 [FGFR1, FGFR3] 1 3 4 1149 - TW 37 [BCL2, BCL2L1] 0 4 4 1259 - BMN-673 [PARP1] 1 3 4 1372 - Trametinib [MAP2K1 (MEK1), MAP2K2 (MEK2)] 3 1 4 152 - CP466722 [ATM] 1 3 4 157 - JNK-9L [JNK] 0 4 4 182 - Obatoclax Mesylate [BCL2, BCL2L1, MCL1] 0 4 4 200 - LAQ824 [HDAC] 0 4 4 254 - AC220 [FLT3] 4 0 4 255 - CP724714 [ERBB2] 3 1 4 266 - Zibotentan, ZD4054 [Endothelin A Receptor] 2 2 4 287 - KIN001-244 [PDPK1 (PDK1)] 2 2 4 310 - YM201636 [FYV1] 2 2 4 345 - KIN001-270 [CDK9] 2 2 4 1004 - Vinblastine [Microtubules] 0 3 3 1005 - Cisplatin [DNA crosslinker] 0 3 3 1010 - Gefitinib [EGFR] 3 0 3 1011 - ABT-263 [BCL2, BCL2L1, BCL2L2] 1 2 3 1026 - 17-AAG [HSP90] 0 3 3 1029 - AMG-706 [VEGFR, RET, c-KIT, PDGFR] 3 0 3 1170 - CCT018159 [HSP90] 0 3 3 1230 - IOX2 [EGLN1] 3 0 3 1236 - UNC0638 [G9a(EHMT2), GLP(EHMT1)] 2 1 3 133 - Doxorubicin [DNA intercalating] 0 3 3 1494 - SN-38 [TOP1] 1 2 3 1495 - AZD-2281 [PARP1, PARP2] 2 1 3 192 - LFM-A13 [BTK] 2 1 3 201 - Epothilone B [Microtubules] 0 3 3 206 - Ruxolitinib [JAK1, JAK2, TYK2] 3 0 3 221 - TAK-715 [p38a] 1 2 3 222 - BX-912 [PDPK1 (PDK1)] 3 0 3 225 - Genentech Cpd 10 [AURKA, AURKB] 2 1 3 226 - GSK1070916 [AURKB] 2 1 3 249 - XL-184 [VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, Tie2,AXL] 2 1 3 252 - WZ3105 [CLK2, CNSK1E, FLT3, ULK1] 1 2 3 260 - NG-25 [MAP3K7 (TAK1)] 3 0 3 268 - YM155 [BIRC5 (Survivin)] 1 2 3 271 - VNLG/124 [HDAC, RAR ] 3 0 3 277 - ABT-869 [VEGFR and PDGFR family] 3 0 3 281 - CH5424802 [ALK] 3 0 3 292 - Masitinib [KIT] 1 2 3 294 - MPS-1-IN-1 [MPS1] 2 1 3 295 - NVP-BHG712 [EPHB4] 3 0 3 298 - OSI-930 [KIT, VEGFR, PDGFR] 1 2 3 30 - Sorafenib [PDGFRA, PDGFRB, KDR, KIT, FLT3] 3 0 3 304 - SB52334 [ALK5] 3 0 3 328 - SNX-2112 [HSP90] 2 1 3 333 - T0901317 [LXR] 2 1 3 346 - THZ-2-102-1 [CDK7] 2 1 3 89 - Parthenolide [NFKB1] 2 1 3 1008 - Methotrexate [Dihydrofolate reductase (DHFR)] 0 2 2 1016 - Temsirolimus [MTOR] 1 1 2 1017 - Olaparib [PARP1, PARP2] 1 1 2 1018 - ABT-888 [PARP1, PARP2] 1 1 2 1019 - Bosutinib [SRC, ABL, TEC] 2 0 2 1028 - VX-702 [p38] 2 0 2 1031 - Elesclomol [HSP70] 1 1 2 1032 - Afatinib [ERBB2, EGFR] 2 0 2 1033 - Vismodegib [SMO] 1 1 2 1036 - PLX4720 [BRAF] 2 0 2 1039 - SL 0101-1 [RSK, AURKB, PIM3] 0 2 2 1046 - 681640 [WEE1, CHEK1] 0 2 2 1060 - PD-0325901 [MAP2K1 (MEK1), MAP2K2 (MEK2)] 2 0 2 1066 - AZD6482 [PI3Kbeta] 0 2 2 1091 - BMS-536924 [IGF1R] 0 2 2 1133 - JNJ-26854165 [MDM2] 0 2 2 1142 - HG-5-113-01 [LOK, LTK, TRCB, ABL(T315I)] 1 1 2 1143 - HG-5-88-01 [EGFR, ADCK4] 1 1 2 1166 - QL-VIII-58 [MTOR, ATR] 0 2 2 119 - Lapatinib [ERBB2, EGFR] 2 0 2 1243 - piperlongumine [Increases ROS levels] 0 2 2 1248 - FK866 [NAMPT] 1 1 2 1264 - SGC0946 [Q8TEK3 (DOT1L)] 2 0 2 136 - Mitomycin C [DNA crosslinker] 1 1 2 1373 - Dabrafenib [BRAF] 1 1 2 140 - Vinorelbine [Microtubules] 0 2 2 147 - NSC-87877 [PTPN6 (SHP-1), PTPN11 (SHP-2)] 2 0 2 1529 - MLN4924 [NEDD8-activating enzyme] 0 2 2 155 - AP-24534 [ABL] 1 1 2 178 - BAY 61-3606 [SYK] 0 2 2 184 - BMS-754807 [IGF1R] 1 1 2 185 - OSI-906 [IGF1R] 2 0 2 194 - AUY922 [HSP90] 0 2 2 231 - FMK [RSK] 1 1 2 261 - TL-1-85 [MAP3K7 (TAK1)] 2 0 2 263 - FR-180204 [ERK] 2 0 2 274 - PXD101, Belinostat [HDAC] 1 1 2 302 - PI-103 [PI3Ka, PRKDC (DNAPK)] 2 0 2 303 - PIK-93 [PI4K, PI3K] 2 0 2 305 - TPCA-1 [IKK] 2 0 2 306 - TG101348 [JAK2] 0 2 2 312 - AV-951 [VEGFR] 2 0 2 38 - AZD-0530 [SRC, ABL1] 2 0 2 45 - Z-LLNle-CHO [g-secretase] 0 2 2 5 - Sunitinib [PDGFRA, PDGFRB, KDR, KIT, FLT3] 2 0 2 60 - BI-2536 [PLK1, PLK2, PLK3] 0 2 2 94 - TGX221 [PI3Kbeta] 2 0 2 1 - Erlotinib [EGFR] 1 0 1 1001 - AICAR [AAPK1 (AMPK) agonist] 0 1 1 1006 - Cytarabine [DNA synthesis] 1 0 1 1007 - Docetaxel [Microtubules] 0 1 1 1020 - Lenalidomide [TNFA] 0 1 1 1022 - AZD7762 [CHEK1, CHEK2] 0 1 1 1023 - GW 441756 [NTRK1] 1 0 1 1037 - BX-795 [TBK1, PDPK1, IKK, AURKB, AURKC] 0 1 1 104 - Bortezomib [Proteasome] 0 1 1 1042 - BIRB 0796 [p38, JNK2] 0 1 1 1061 - SB590885 [BRAF] 1 0 1 1114 - Cetuximab [EGFR] 1 0 1 1161 - ZG-10 [IRAK1] 0 1 1 1219 - PFI-1 [BRD2, BRD3, BRD4] 0 1 1 134 - Etoposide [TOP2] 1 0 1 135 - Gemcitabine [DNA replication] 1 0 1 1371 - PLX4720 (rescreen) [BRAF] 1 0 1 1375 - Temozolomide [DNA akylating agent] 0 1 1 1377 - Afatinib (rescreen) [ERBB2, EGFR] 1 0 1 1527 - GDC0941 (rescreen) [PI3K] 1 0 1 159 - HG-6-64-1 [BRAFV600E, TAK, MAP4K5] 1 0 1 166 - FTI-277 [Farnesyl transferase (FNTA)] 1 0 1 167 - OSU-03012 [PDPK1 (PDK1)] 0 1 1 171 - AKT inhibitor VIII [AKT1, AKT2, AKT3] 0 1 1 172 - Embelin [XIAP] 0 1 1 176 - IPA-3 [PAK1, PAK2, PAK3] 0 1 1 180 - Thapsigargin [sarco-endoplasmic reticulum Ca2+-ATPases] 0 1 1 186 - Bexarotene [Retinioic acid X family agonist] 1 0 1 193 - GW-2580 [CSF1R (cFMS)] 1 0 1 197 - Bryostatin 1 [PRKC] 1 0 1 199 - Pazopanib [VEGFR, PDGFRA, PDGFRB, KIT] 1 0 1 203 - BMS-345541 [IKBKB] 1 0 1 204 - Tipifarnib [Farnesyl-transferase (FNTA)] 0 1 1 207 - AS601245 [JNK ] 0 1 1 211 - TL-2-105 [CRAF] 1 0 1 219 - AT-7519 [CDK9] 1 0 1 223 - ZSTK474 [PI3K] 1 0 1 228 - KIN001-102 [AKT1] 1 0 1 229 - LY317615 [PRKCB (PKCbeta)] 0 1 1 238 - CAL-101 [PI3Kdelta] 1 0 1 245 - UNC0638 [G9a(EHMT2), GLP(EHMT1)] 0 1 1 253 - XMD14-99 [EPHB3, CAMK1] 1 0 1 256 - JW-7-24-1 [LCK] 1 0 1 258 - STF-62247 [stimulates autophagy] 1 0 1 262 - VX-11e [ERK] 1 0 1 265 - Tubastatin A [HDAC6] 1 0 1 273 - CUDC-101 [HDAC, EGFR] 1 0 1 275 - I-BET [BRD2, BRD3, BRD4] 1 0 1 276 - CAY10603 [HDAC6] 1 0 1 279 - BIX02189 [MAP2K5 (MEK5)] 1 0 1 282 - EKB-569 [EGFR] 0 1 1 283 - GSK2126458 [PI3K, MTOR] 1 0 1 286 - KIN001-236 [TIE2] 1 0 1 288 - KIN001-055 [JAK3, MNK1] 1 0 1 29 - AZ628 [BRAF] 1 0 1 291 - KIN001-266 [MAP3K8 (COT)] 1 0 1 299 - OSI-027 [MTORC1/2] 1 0 1 3 - Rapamycin [MTOR] 1 0 1 301 - PHA-793887 [CDK-pan] 1 0 1 308 - XL-880 [MET] 0 1 1 309 - Y-39983 [ROCK] 0 1 1 32 - VX-680 [AURKA, AURKB, AURKC, FLT3, ABL1, JAK2] 1 0 1 329 - QL-XI-92 [DDR1] 0 1 1 331 - QL-X-138 [MNK2, PRKDC (DNAPK), MTOR, BTK, JAK3] 1 0 1 332 - XMD15-27 [CAMK2B, CLK2, DYRK1A, MAST1, STK39] 1 0 1 34 - Imatinib [ABL, KIT, PDGFR] 1 0 1 341 - EX-527 [SIRT1] 1 0 1 344 - THZ-2-49 [CDK9] 1 0 1 37 - Crizotinib [MET, ALK] 1 0 1 51 - Dasatinib [ABL, SRC, KIT, PDGFR] 1 0 1 52 - GNF-2 [ABL [T315I]] 1 0 1 53 - CGP-60474 [CDK1,CDK2,CDK5,CDK7,CDK9] 0 1 1 55 - A-770041 [SRC family] 1 0 1 56 - WH-4-023 [SRC family, ABL] 1 0 1 59 - WZ-1-84 [BMX] 1 0 1 63 - BMS-509744 [ITK] 1 0 1 71 - Pyrimethamine [Dihydrofolate reductase (DHFR)] 1 0 1 86 - A-443654 [AKT1, AKT2, AKT3] 0 1 1 87 - GW843682X [PLK1] 0 1 1 9 - MG-132 [Proteasome] 0 1 1